TABLE 1

Suzetrigine prescribing and cost information

IndicationApproved by US Food and Drug Administration to treat acute postoperative pain for 14 days
DoseLoading: 100 mg
Maintenance: 50 mg every 12 hours
DurationHalf-life of 23.6 hours
Cost$15.50 per pill18 (typical course is 2 weeks)
Common side effectsNausea and vomiting, pruritis, rash, muscle spasms, increased serum creatine phosphokinase level
ContraindicationsHormonal contraceptives: may impair efficacy
Cirrhosis: reduce dose for Child-Pugh class B; do not use in Child-Pugh class C
CYP3A substrates: inhibitors may cause accumulation of drug and metabolites; inducers may reduce effect
  • Based on information from reference 11.